CRKL binding to BCR-ABL and BCR-ABL transformation

Leuk Lymphoma. 1999 Mar;33(1-2):119-26. doi: 10.3109/10428199909093732.

Abstract

The SH2-SH3 domain-containing adaptor protein CRKL is the predominant tyrosine phosphorylated protein in chronic myelogenous leukemia (CML) neutrophils and BCR-ABL-expressing cell lines. The amino terminal CRKL SH3 domain binds directly to a proline-rich region in the C-terminus of BCR-ABL. BCR-ABL mutants with deletions of this region were constructed to assess biologic effects of eliminating the CRKL binding site. Yeast two-hybrid analysis and gel overlay assays show eradication of the direct interaction of CRKL with BCR-ABL in the proline deletion mutants. However, these BCR-ABL mutants transform myeloid cells to growth factor independence, and in these cells CRKL is tyrosine phosphorylated and associates with BCR-ABL. These findings suggest both direct and indirect interactions of CRKL with BCR-ABL. Thus, disruption of the direct interaction with BCR-ABL has not excluded a role for CRKL in BCR-ABL-mediated transformation.

MeSH terms

  • Adaptor Proteins, Signal Transducing*
  • Binding Sites / genetics
  • Cell Transformation, Neoplastic / genetics
  • Cell Transformation, Neoplastic / metabolism*
  • Cells, Cultured
  • Fusion Proteins, bcr-abl / genetics
  • Fusion Proteins, bcr-abl / metabolism*
  • Humans
  • K562 Cells
  • Mutagenesis, Site-Directed
  • Nuclear Proteins / chemistry
  • Nuclear Proteins / metabolism*
  • Phosphorylation
  • Proline / genetics
  • Proline / physiology
  • Protein Binding / genetics
  • Sequence Deletion / genetics
  • Transfection
  • Tyrosine / metabolism

Substances

  • Adaptor Proteins, Signal Transducing
  • CRKL protein
  • Nuclear Proteins
  • Tyrosine
  • Proline
  • Fusion Proteins, bcr-abl