I(ARC), a novel arachidonate-regulated, noncapacitative Ca(2+) entry channel

J Biol Chem. 2000 Mar 31;275(13):9114-9. doi: 10.1074/jbc.275.13.9114.

Abstract

Along with the inositol trisphosphate-induced release of stored Ca(2+), a receptor-enhanced entry of Ca(2+) is a critical component of intracellular Ca(2+) signals generated by agonists acting at receptors coupled to the activation of phospholipase C. Although the simple emptying of the intracellular Ca(2+) stores is known to be capable of activating Ca(2+) entry via the so-called "capacitative" mechanism, recent evidence suggests that Ca(2+) entry at physiological agonist concentrations, where oscillatory Ca(2+) signals are typically observed, does not conform to such a model. Instead, a noncapacitative Ca(2+) entry pathway regulated by arachidonic acid appears to be responsible for Ca(2+) entry under these conditions. Using whole-cell patch clamp techniques we demonstrate that low concentrations of arachidonic acid activate a Ca(2+)-selective current that is superficially similar to the store-operated current I(CRAC), but which also demonstrates certain distinct features. We have named this novel current I(ARC) (for arachidonate-regulated calcium current). Importantly, I(ARC) can be readily activated in cells whose Ca(2+) stores have been maximally depleted. I(ARC) represents a novel Ca(2+) entry pathway that is entirely separate from those activated by store depletion and is specifically activated at physiological levels of stimulation.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Arachidonic Acid / pharmacology*
  • Calcium / metabolism*
  • Calcium Channel Agonists / pharmacology*
  • Calcium Channels / metabolism*
  • Cell Line
  • Humans
  • Ion Transport
  • Membrane Potentials

Substances

  • Calcium Channel Agonists
  • Calcium Channels
  • Arachidonic Acid
  • Calcium