Highly efficient synthesis of 1-thioglycosides in solution and solid phase using iminophosphorane bases

Carbohydr Res. 2000 Apr 20;325(3):169-76. doi: 10.1016/s0008-6215(99)00327-4.

Abstract

Disaccharides of 1-thioglycosides, an important class of glycomimics, can be synthesized by direct S-alkylation in exceptionally high yields when iminophosphorane bases are employed. The reaction conditions employed appear to be general and stereospecific. Axial and equatorial 4-triflates and primary tosylates of alkyl pyranosides provided excellent yields of thio-disaccharides without substantial elimination products. The iminophosphorane bases also proved to be useful in solid support-bound couplings of thioglycosides though with lower efficiency.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alkylation
  • Chromatography, High Pressure Liquid
  • Phosphoranes / chemistry*
  • Thioglycosides / chemical synthesis*

Substances

  • Phosphoranes
  • Thioglycosides