An essential intermediate in the folding of dihydrofolate reductase

Proc Natl Acad Sci U S A. 2000 May 23;97(11):5866-70. doi: 10.1073/pnas.100547697.

Abstract

The folding of Escherichia coli dihydrofolate reductase was examined at pH 7.8 and 15 degrees C by using stopped-flow fluorescence and absorbance spectroscopies. The formation of a highly fluorescent intermediate occurs with relaxation times ranging between 142 and 343 msec, whereas stopped-flow absorbance spectroscopy using methotrexate binding assays shows a distinct lag phase during these time frames for the native state. The lag in absorbance kinetics and the lack of fast-track folding events indicate that the formation of this ensemble of intermediates is an obligatory step in the folding reaction.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Bacterial Proteins / chemistry*
  • Bacterial Proteins / metabolism
  • Escherichia coli / enzymology
  • Methotrexate / metabolism
  • Models, Molecular
  • Protein Binding
  • Protein Conformation
  • Protein Folding
  • Spectrometry, Fluorescence
  • Tetrahydrofolate Dehydrogenase / chemistry*
  • Tetrahydrofolate Dehydrogenase / metabolism

Substances

  • Bacterial Proteins
  • Tetrahydrofolate Dehydrogenase
  • Methotrexate