A Simple One-Pot Procedure for the Direct Conversion of Alcohols to Azides via Phosphate Activation

Org Lett. 2000 Jun 29;2(13):1959-1961. doi: 10.1021/ol0060376.

Abstract

A one-pot procedure was developed to prepare efficiently alkyl azides from alkanols using bis(2,4-dichlorophenyl) phosphate activation. 4-(Dimethylamino)pyridine was used as a base, and phosphorylpyridinium azide is believed to be the activating agent under this condition.