Effect of protein kinase A on calcium sensitivity of force and its sarcomere length dependence in human cardiomyocytes

Cardiovasc Res. 2000 Jun;46(3):487-95. doi: 10.1016/s0008-6363(00)00050-x.

Abstract

Objective: We investigated whether the Frank-Starling mechanism is absent or preserved in end-stage failing human myocardium and if phosphorylation of contractile proteins modulates its magnitude through the sarcomere length-dependence of calcium sensitivity of isometric force development.

Methods: The effect of phosphorylation of troponin I and C-protein by the catalytic subunit of protein kinase A (3 microg/ml; 40 min at 20 degrees C) was studied in single Triton-skinned human cardiomyocytes isolated from donor and end-stage failing left ventricular myocardium at sarcomere lengths measured at rest of 1.8, 2.0 and 2.2 microm. Isometric force development was studied at various free-calcium concentrations before and after protein kinase A incubation at 15 degrees C (pH 7.1).

Results: Maximal isometric tension at 2.2 microm amounted to 39.6+/-10.4 and 33.7+/-3.5 kN/m2 in donor and end-stage failing cardiomyocytes, respectively. The midpoints of the calcium sensitivity curves (pCa50) of donor and end-stage failing hearts differed markedly at all sarcomere lengths (mean delta pCa50=0.22). A reduction in sarcomere length from 2.2 to 1.8 microm caused reductions in maximum isometric force to 64% and 65% and in pCa50 by 0.10 and 0.08 pCa units in donor and failing cardiomyocytes, respectively. In donor tissue, the effect of protein kinase A treatment was rather small, while in end-stage failing myocardium it was much larger (delta pCa50=0.24) irrespective of sarcomere length.

Conclusions: The data obtained indicate that the Frank-Starling mechanism is preserved in end-stage failing myocardium and suggest that sarcomere length dependence of calcium sensitivity and the effects of phosphorylation of troponin I and C-protein are independent.

MeSH terms

  • Calcium / metabolism*
  • Carrier Proteins / metabolism
  • Cyclic AMP-Dependent Protein Kinases / pharmacology*
  • Heart Failure / metabolism*
  • Humans
  • In Vitro Techniques
  • Isometric Contraction*
  • Myocardium / cytology
  • Myocardium / metabolism*
  • Phosphorylation
  • Sarcomeres / drug effects*
  • Troponin I / metabolism

Substances

  • Carrier Proteins
  • Troponin I
  • citrate-binding transport protein
  • Cyclic AMP-Dependent Protein Kinases
  • Calcium