Ristocetin-dependent, but not botrocetin-dependent, binding of von Willebrand factor to the platelet glycoprotein Ib-IX-V complex correlates with shear-dependent interactions

Blood. 2001 Jan 1;97(1):162-8. doi: 10.1182/blood.v97.1.162.

Abstract

Under conditions of high shear stress, both hemostasis and thrombosis are initiated by the interaction of the platelet membrane glycoprotein (GP) Ib-IX-V complex with its adhesive ligand, von Willebrand factor (vWF), in the subendothelial matrix or plasma. This interaction involves the A1 domain of vWF and the N-terminal extracellular region of GP Ibalpha (His-1-Glu-282), and it can also be induced under static conditions by the modulators ristocetin and botrocetin. In this study, a panel of anti-vWF and anti-GP Ibalpha antibodies-previously characterized for their effects on ristocetin- and botrocetin-dependent vWF-GP Ib-IX-V interactions-was analyzed for their capacity to inhibit either the adhesion of Chinese hamster ovary cells expressing recombinant GP Ibalpha to surface-associated vWF under hydrodynamic flow or shear-stress-induced platelet aggregation. The combined results suggest that the shear-dependent interactions between vWF and GP Ibalpha closely correlate with ristocetin- rather than botrocetin-dependent binding under static conditions and that certain anti-vWF monoclonal antibodies are able to selectively inhibit shear-dependent platelet aggregation.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Antibodies, Monoclonal / pharmacology
  • Blood Viscosity
  • Crotalid Venoms / pharmacology
  • Dose-Response Relationship, Drug
  • Epitopes
  • Humans
  • Models, Molecular
  • Platelet Adhesiveness / drug effects
  • Platelet Aggregation / drug effects
  • Platelet Glycoprotein GPIb-IX Complex / immunology
  • Platelet Glycoprotein GPIb-IX Complex / metabolism
  • Protein Binding / drug effects
  • Protein Structure, Tertiary
  • Ristocetin / pharmacology*
  • Stress, Mechanical
  • von Willebrand Factor / drug effects*
  • von Willebrand Factor / immunology
  • von Willebrand Factor / metabolism

Substances

  • Antibodies, Monoclonal
  • Crotalid Venoms
  • Epitopes
  • Platelet Glycoprotein GPIb-IX Complex
  • von Willebrand Factor
  • Ristocetin
  • botrocetin