Expression of multidrug resistance-related markers in gastric cancer

Anticancer Res. 2000 Nov-Dec;20(6C):4809-14.

Abstract

Background: To detect the expression of glutathione S-transferase Pi(GST-pi), multidrug resistance-associated protein (MRP), lung-resistance protein(LRP), multidrug resistance gene1 (MDR1) and MGr1 antigen(MGr1-Ag) in the patients with primary gastric cancer and without any prior chemotherapy and to evaluate the correlations between them.

Patients and methods: The expression of GST-pi, MRP, LRP and MDR1 in cancer tissue and the adjacent non-cancerous tissue from 50 patients was examined by semiquantitative reverse transcription-polymerase chain reaction (RT-PCR). The expression of MGr1-Ag in these tissues was also examined by immunohistochemistry.

Results: The positive rate of GST-pi mRNA, MRP mRNA, LRP mRNA, MDR1mRNA and MGr1-Ag in gastric cancer tissue was 36.00%, 12.00%, 10.00%, 10.00% and 18.00% respectively. The overall positive rate of their expression was 58.00%. Clinicopathological factors were not significantly related to their expression. No significant correlation was observed between these markers.

Conclusion: These MDR markers are differently over-expressed and no coexpression exists in gastric cancer. MGr1-Ag was a novel MDR protein.

MeSH terms

  • ATP Binding Cassette Transporter, Subfamily B, Member 1 / analysis
  • ATP Binding Cassette Transporter, Subfamily B, Member 1 / genetics
  • Adenocarcinoma / genetics*
  • Adenocarcinoma / pathology
  • DNA Primers
  • Drug Resistance, Multiple*
  • Female
  • Glutathione Transferase / analysis
  • Glutathione Transferase / genetics
  • Humans
  • Immunohistochemistry
  • Male
  • Middle Aged
  • Neoplasm Proteins / analysis
  • Neoplasm Proteins / genetics
  • Reverse Transcriptase Polymerase Chain Reaction
  • Stomach Neoplasms / genetics*
  • Stomach Neoplasms / pathology
  • Transcription, Genetic
  • Vault Ribonucleoprotein Particles / genetics

Substances

  • ATP Binding Cassette Transporter, Subfamily B, Member 1
  • DNA Primers
  • Neoplasm Proteins
  • Vault Ribonucleoprotein Particles
  • major vault protein
  • Glutathione Transferase