The effect of gamma-vinyl-GABA on the consumption of concurrently available oral cocaine and ethanol in the rat

Pharmacol Biochem Behav. 2001 Feb;68(2):291-9. doi: 10.1016/s0091-3057(00)00456-1.

Abstract

It has frequently been reported that a high percentage of individuals, identified as either alcohol- or cocaine-dependent, concurrently abuse both drugs. The experiments reported here represent a continuing effort to develop an animal model to predict the effects of a potential pharmacotherapeutic agent on concurrently available oral ethanol and cocaine. These experiments utilized drinkometer circuitry to assess the effects of gamma-vinyl-GABA (GVG), a gamma-aminobutyric acid (GABA) transaminase inhibitor, on the consumption and temporal pattern of responses for orally self-administered ethanol and cocaine. The results of these experiments showed that GVG, at doses of 100, 200 and 300 mg/kg, reduced both ethanol and cocaine consumption in a dose-related manner. When compared to vehicle, GVG at all doses significantly reduced ethanol consumption while consumption of cocaine was significantly reduced only at 300 mg/kg. This is consistent with data showing that GVG reduces consumption of these drugs when administered alone and data showing that GVG is more potent in reducing ethanol-induced compared to cocaine-induced extracellular dopamine in the nucleus accumbens. Analysis of the temporal pattern of drinking across the session suggests that GVG's effects are due to a disruption of the reinforcing properties of ethanol and cocaine rather than a more general reduction in motor behavior. These data suggest that GVG has potential for clinical use in populations that abuse either alcohol or cocaine alone or in combination.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Alcohol Drinking / drug therapy*
  • Animals
  • Behavior, Addictive / drug therapy
  • Cocaine / analogs & derivatives*
  • Cocaine / blood
  • Cocaine-Related Disorders / drug therapy*
  • Disease Models, Animal*
  • Dose-Response Relationship, Drug
  • Enzyme Inhibitors / therapeutic use*
  • Male
  • Rats
  • Rats, Wistar
  • Self Administration
  • Vigabatrin / therapeutic use*

Substances

  • Enzyme Inhibitors
  • benzoylecgonine
  • Vigabatrin
  • Cocaine