Hepatocyte Growth Factor/scatter factor-induces phosphorylation of cortactin in A431 cells in a Src kinase-independent manner

Oncogene. 2001 Jun 21;20(28):3735-45. doi: 10.1038/sj.onc.1204474.

Abstract

The Hepatocyte Growth Factor receptor transduces proliferating and scattering signals in epithelial and endothelial cells. We have explored potential interactions of the HGF/SF receptor beta-subunit (p145(beta MET)) with F-actin binding partners aiming to identify novel downstream effectors implicated in HGF/SF pluripotent signalling. Cortactin, a p80/85 F-actin binding protein, was found phosphorylated on tyrosine in response to HGF-SF in A431 human epidermoid carcinoma cells, expressing the HGF/SF receptor (c-MET). The HGF/SF receptor was enriched in the detergent-insoluble fraction and was found to co-precipitate with cortactin and to associate in vitro with cortactin. The Grb2 small adapter protein known to associate via its Src homology 2 domain (SH2) with the MET C-terminus, was also associated with cortactin. Transient transfection of A431 cells with dominant-negative Grb2 constructs has revealed that the Grb2-C-SH3 domain possesses a central role in cortactin phosphorylation in response to HGF/SF. Finally, tyrosine phosphorylation of cortactin was found uncoupled of endogenous c-Src kinase activity, thus further supporting the hypothesis that cortactin is a direct target of the MET kinase. We propose that cortactin may constitute a docking site for MET-derived signals within the cytoskeleton.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adaptor Proteins, Signal Transducing*
  • CSK Tyrosine-Protein Kinase
  • Cell Fractionation
  • Cortactin
  • Cytoskeleton / metabolism
  • Detergents
  • GRB2 Adaptor Protein
  • Hepatocyte Growth Factor / metabolism*
  • Hepatocytes
  • Humans
  • Microfilament Proteins / metabolism*
  • Octoxynol
  • Phosphorylation
  • Protein-Tyrosine Kinases / metabolism*
  • Proteins / genetics
  • Proteins / metabolism
  • Proto-Oncogene Proteins c-met / metabolism
  • Tumor Cells, Cultured
  • Tyrosine / metabolism
  • src Homology Domains
  • src-Family Kinases

Substances

  • Adaptor Proteins, Signal Transducing
  • CTTN protein, human
  • Cortactin
  • Detergents
  • GRB2 Adaptor Protein
  • GRB2 protein, human
  • Microfilament Proteins
  • Proteins
  • Tyrosine
  • Hepatocyte Growth Factor
  • Octoxynol
  • Protein-Tyrosine Kinases
  • Proto-Oncogene Proteins c-met
  • CSK Tyrosine-Protein Kinase
  • src-Family Kinases
  • CSK protein, human