Absorption and preferential vagina-to-uterus distribution after vaginal administration of (99m)Tc-pertechnetate in postmenopausal women

Fertil Steril. 2001 Dec;76(6):1108-12. doi: 10.1016/s0015-0282(01)02905-3.

Abstract

Objective: To investigate in vivo and in humans the mechanisms and kinetics of vagina-to-uterus distribution.

Design: Controlled clinical study.

Setting: Volunteers in an academic research environment.

Patient(s): Six postmenopausal women undergoing transabdominal hysterectomy were selected.

Intervention(s): Women received 0.2 mL of (99m)Tc-pertechnetate vaginally. In three patients the cervical canal was previously sealed by means of surgical glue. Six postmenopausal women who had received (99m)Tc-pertechnetate intravenously for a thyroid scintigraphy were considered as a control.

Main outcome measure(s): Radioactivity was assessed every 30 minutes for 6 hours in the pelvis and in body regions where (99m)Tc-pertechnetate normally accumulates (thyroid, salivary glands, and stomach).

Result(s): Uterine activity appeared after 60 minutes and peaked between 120 to 210 minutes. These same times were observed in the patients who had a sealed cervix. Thyroid uptake appeared after 180 minutes and peaked between 210 and 330 minutes. Uterine uptake did not occur in any of the intravenous patients; their thyroid uptake was rapid, appearing after 30 minutes.

Conclusion(s): Preferential vagina-to-uterus distribution, at least in postmenopausal women, is not simply due an intracanalicular passage but is mediated by absorption of substances and probably by a countercurrent transfer mechanism.

Publication types

  • Clinical Trial
  • Controlled Clinical Trial

MeSH terms

  • Absorption
  • Administration, Intravaginal
  • Female
  • Humans
  • Pilot Projects
  • Postmenopause
  • Radionuclide Imaging
  • Radiopharmaceuticals / administration & dosage
  • Radiopharmaceuticals / pharmacokinetics*
  • Salivary Glands / diagnostic imaging
  • Sodium Pertechnetate Tc 99m / administration & dosage
  • Sodium Pertechnetate Tc 99m / pharmacokinetics*
  • Stomach / diagnostic imaging
  • Thyroid Gland / diagnostic imaging
  • Uterus / diagnostic imaging
  • Uterus / metabolism*
  • Vagina / diagnostic imaging
  • Vagina / drug effects
  • Vagina / metabolism*

Substances

  • Radiopharmaceuticals
  • Sodium Pertechnetate Tc 99m