Transdermal contraception: evaluation of three transdermal norelgestromin/ethinyl estradiol doses in a randomized, multicenter, dose-response study

Am J Obstet Gynecol. 2002 Jan;186(1):15-20. doi: 10.1067/mob.2002.118844.

Abstract

Objective: The objective of this study was to identify the dose for a contraceptive patch that provides a predetermined level of ovulation suppression and cycle control and that is well tolerated.

Study design: In this randomized study, 610 subjects received 10-, 15-, or 20-cm(2) patch dose sizes (20-cm(2), Ortho Evra/Evra) (Janssen Pharmaceutica, NV Belgium) or Ortho-Cyclen/Cilest (Janssen Pharmaceutica, NV Belgium) for up to 4 cycles. As with Ortho-Cyclen, patch regimens included 21 dosing days (3 consecutive 7-day patches) followed by 1 dose-free week.

Results: The patch regimens demonstrated a dose-response for ovulation suppression and cycle control. Presumed ovulation, determined on the basis of serum progesterone concentrations > or = 3 ng/mL in cycles 1 and 3, occurred in 6.2% (Ortho Evra) and 7.2% (Ortho-Cyclen) of subjects. At cycle 3, breakthrough bleeding/spotting was reported by 10.5% and 15.0% of subjects, respectively. Compliance with each patch was superior to that with Ortho-Cyclen (all P <.001). All regimens had safety profiles typical of oral contraceptives.

Conclusion: The 20-cm(2) patch (Ortho Evra) provided ovulation suppression, cycle control, and safety similar to that of Ortho-Cyclen, with significantly better compliance.

Publication types

  • Clinical Trial
  • Multicenter Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Cutaneous
  • Adult
  • Contraceptive Agents, Female / administration & dosage*
  • Contraceptive Agents, Female / adverse effects
  • Contraceptive Agents, Female / pharmacology
  • Dose-Response Relationship, Drug
  • Estradiol / blood
  • Estradiol Congeners / administration & dosage*
  • Estradiol Congeners / adverse effects
  • Estradiol Congeners / pharmacology
  • Ethinyl Estradiol / administration & dosage*
  • Ethinyl Estradiol / adverse effects
  • Ethinyl Estradiol / pharmacology
  • Female
  • Humans
  • Luteinizing Hormone / blood
  • Menstrual Cycle / drug effects
  • Ovary / metabolism
  • Ovulation
  • Patient Compliance
  • Pituitary Gland / metabolism
  • Safety

Substances

  • Contraceptive Agents, Female
  • Estradiol Congeners
  • Ethinyl Estradiol
  • Estradiol
  • Luteinizing Hormone