Calpain is a signal transducer and activator of transcription (STAT) 3 and STAT5 protease

Blood. 2002 Mar 1;99(5):1850-2. doi: 10.1182/blood.v99.5.1850.

Abstract

Truncation of signal transducer and activator of transcription (STAT) 5 at the carboxy-terminal domain, either by genetic engineering or by proteolytic cleavage, results in generation of dominant-negative forms. A nuclear serine protease expressed in the myeloid precursor cells is known to mediate this cleavage, but other proteases responsible for this reaction were unknown. We found that calpain, a ubiquitously expressed cysteine protease, also trims STAT5 in vivo and in vitro, within the carboxy-terminal domain. Nuclear element is not necessary for calpain-mediated STAT5 cleavage, since this process occurs in platelets. We also found that STAT3 is a substrate for calpain in vivo and in vitro, indicating that calpain-mediated cleavage is a common feature of STAT3 and STAT5. Thus, our study reveals a novel pathway for posttranslational modification of STAT3 and STAT5.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Blood Platelets / enzymology
  • Calpain / metabolism
  • Calpain / pharmacology
  • Calpain / physiology*
  • Cysteine Endopeptidases / metabolism
  • Cysteine Endopeptidases / pharmacology
  • Cysteine Endopeptidases / physiology
  • DNA-Binding Proteins / isolation & purification
  • DNA-Binding Proteins / metabolism
  • Enzyme Activation
  • Humans
  • Milk Proteins*
  • Protein Processing, Post-Translational / drug effects
  • STAT3 Transcription Factor
  • STAT5 Transcription Factor
  • Signal Transduction
  • Trans-Activators / isolation & purification
  • Trans-Activators / metabolism

Substances

  • DNA-Binding Proteins
  • Milk Proteins
  • STAT3 Transcription Factor
  • STAT3 protein, human
  • STAT5 Transcription Factor
  • Trans-Activators
  • Calpain
  • Cysteine Endopeptidases