Regulation of ROMK channels by protein tyrosine kinase and tyrosine phosphatase

Trends Cardiovasc Med. 2002 Apr;12(3):138-42. doi: 10.1016/s1050-1738(02)00155-x.

Abstract

Renal outer medulla K (ROMK) channels play an important role in K recycling in the thick ascending limb and in K secretion in the cortical collecting duct. ROMK1, a member of the ROMK family, has been shown to be a substrate for protein tyrosine kinase (PTK). The tyrosine phosphorylation of ROMK channels increases with low dietary K intake and decreases with high dietary K intake. Moreover, the stimulation of tyrosine phosphorylation of ROMK1 channels decreases the number of K channels by facilitating endocytosis. In contrast, the stimulation of tyrosine dephosphorylation increases the number of ROMK1 channels in the cell membrane by enhancing membrane insertion. PTK and tyrosine phosphatase-induced regulation of ROMK1 channels play a key role in mediating the effect of the dietary K intake on renal K secretion.

Publication types

  • Research Support, U.S. Gov't, P.H.S.
  • Review

MeSH terms

  • Animals
  • Enzyme Activation / drug effects
  • Humans
  • Kidney / drug effects*
  • Kidney / metabolism
  • Potassium / metabolism
  • Potassium Channels / metabolism*
  • Potassium Channels, Inwardly Rectifying*
  • Potassium, Dietary / pharmacology*
  • Protein Tyrosine Phosphatases / metabolism*
  • Protein-Tyrosine Kinases / metabolism*

Substances

  • KCNJ1 protein, human
  • Potassium Channels
  • Potassium Channels, Inwardly Rectifying
  • Potassium, Dietary
  • Protein-Tyrosine Kinases
  • Protein Tyrosine Phosphatases
  • Potassium