125I-iomazenil-benzodiazepine receptor binding during psychological stress in rats

Ann Nucl Med. 2002 May;16(3):231-5. doi: 10.1007/BF02996307.

Abstract

Objective: We investigated the changes in 125I-iomazenil (125I-IMZ) benzodiazepine receptor (BZR) binding with psychological stress in a rat model.

Methods: Six male Wistar rats were placed under psychological stress for 1 hour by using a communication box. No physical stress was not received. 1.85 MBq of 125I-IMZ was injected into the lateral tail vein and the rat was killed 3 hours later. Twenty-micrometer-thick sections of the brain were collected and % injected dose per body weight (%ID/BW) of eleven regions (frontal, parietal, temporal, occipital cortices, caudate putamen, accumubens nuclei, globus pallidus, amygdala, thalamus, hippocampus and hypothalamus) were calculated by autoradiography. The %ID/BW of rats which were placed under psychological stress was compared with that of 6 control rats.

Results: The %ID/BW of rats which were placed under psychological stress diffusely tended to show a reduction in 125I-IMZ-BZR binding. A significant decrease in BZR binding was observed in the hippocampus of the rats which were placed under psychological stress.

Conclusion: 125I-IMZ-BZR binding tended to decrease throughout the brain.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Brain / diagnostic imaging
  • Brain / metabolism*
  • Electroshock / adverse effects*
  • Flumazenil / analogs & derivatives*
  • Flumazenil / pharmacokinetics*
  • Male
  • Radionuclide Imaging
  • Radiopharmaceuticals / pharmacokinetics
  • Rats
  • Rats, Wistar
  • Receptors, GABA-A / metabolism*
  • Reference Values
  • Stress, Psychological / diagnostic imaging
  • Stress, Psychological / etiology*
  • Stress, Psychological / metabolism*

Substances

  • Radiopharmaceuticals
  • Receptors, GABA-A
  • Flumazenil
  • iomazenil