Leptin induces mitogenic effect on human choriocarcinoma cell line (JAr) via MAP kinase activation in a glucose-dependent fashion

Placenta. 2003 Apr;24(4):385-91. doi: 10.1053/plac.2002.0905.

Abstract

Leptin and glucose effect on cell growth has been investigated in the JAr human choriocarcinoma cells. When JAr cells were cultured in the presence of 6m M glucose (LG), proliferation and thymidine incorporation were induced by serum but not by leptin. At variance, at 25m M glucose (HG), proliferation and thymidine incorporation were stimulated by leptin and serum to a comparable extent. HG culturing also enhanced leptin-stimulated insulin receptor substrate 1 (IRS1) and MAPK phosphorylation. Blockage of MAPK activity with PD98059 caused an inhibition of glucose- and leptin-dependent thymidine incorporation. At variance with HG conditions no effects were observed in cells cultured in 6m M glucose upon treatment with PD98059. Neither glucose nor leptin determined a modification in leptin receptors total content. In this study, we provide evidence that in placental cells, leptin, similarly to that observed with insulin, stimulates cell proliferation by inducing the IRS1/MAPK pathway in a glucose-dependent fashion.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cell Division / drug effects
  • Choriocarcinoma
  • DNA / biosynthesis
  • Dose-Response Relationship, Drug
  • Drug Combinations
  • Enzyme Inhibitors / pharmacology
  • Female
  • Flavonoids / pharmacology
  • Glucose / pharmacology*
  • Growth Substances / pharmacology*
  • Humans
  • Leptin / pharmacology*
  • Mitogen-Activated Protein Kinases / antagonists & inhibitors
  • Mitogen-Activated Protein Kinases / biosynthesis*
  • Signal Transduction
  • Trophoblasts / drug effects*
  • Trophoblasts / enzymology
  • Trophoblasts / pathology
  • Tumor Cells, Cultured / drug effects
  • Uterine Neoplasms
  • Viral Proteins / metabolism

Substances

  • Drug Combinations
  • Enzyme Inhibitors
  • Flavonoids
  • Growth Substances
  • Leptin
  • TRS1 protein, Human herpesvirus 5
  • Viral Proteins
  • DNA
  • Mitogen-Activated Protein Kinases
  • Glucose
  • 2-(2-amino-3-methoxyphenyl)-4H-1-benzopyran-4-one