3-Diazopyrroles. Part 5 (1). Antibacterial activity of 3-diazo-2-phenylpyrroles

Farmaco. 1992 Dec;47(12):1555-62.

Abstract

3-Diazo-2-phenylpyrroles 3a-g showed antimicrobial activity against Gram-positive bacteria, whereas against Gram-negative strains the inhibitory activity is limited to derivatives 3a and 3c. The substituents at 4 and 5 positions strongly influence the inhibitory activity, but the presence of the diazo group is crucial for appearance of activity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anti-Bacterial Agents / chemical synthesis*
  • Anti-Bacterial Agents / pharmacology
  • Chemical Phenomena
  • Chemistry, Physical
  • Escherichia coli / drug effects
  • Magnetic Resonance Spectroscopy
  • Microbial Sensitivity Tests
  • Pyrroles / chemical synthesis*
  • Pyrroles / pharmacology
  • Spectrophotometry, Ultraviolet
  • Streptomyces / drug effects

Substances

  • Anti-Bacterial Agents
  • Pyrroles