Binding of the benzodiazepine ligand [3H]-RO 15-1788 to membrane preparations of the rabbit and turtle retina

Comp Biochem Physiol C Comp Pharmacol Toxicol. 1992 Feb;101(2):337-42. doi: 10.1016/0742-8413(92)90284-e.

Abstract

1. We have studied the binding of [3H]-RO 15-1788 to membrane preparations of the retina of rabbit (Lepus cunicula) and turtle (Pseudemys scripta elegans). 2. In both species, [3H]-RO 15-1788 binding was maximal at 0 degrees C and decreased with increasing temperature. It was saturable, protein concentration-dependent and specific. Flunitrazepam, unlabelled RO 15-1788 and ethyl-beta-carboline were the most effective displacers, whereas RO 5,4864 was ineffective. 3. In both turtle and rabbit retina, Scatchard analysis indicated the presence of a single binding site for [3H]-RO 15-1788. The KD was 0.75 nM in both turtle and rabbit, while the Bmax were 520 and 250 fmol/mg protein in turtle and rabbit respectively. A study of the association rate of [3H]-RO 15-1788 binding revealed faster kinetics in turtle, as compared to rabbit.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Binding, Competitive
  • Cell Membrane / metabolism
  • Flumazenil / metabolism*
  • Rabbits / metabolism*
  • Receptors, GABA-A / metabolism*
  • Retina / metabolism*
  • Species Specificity
  • Temperature
  • Turtles / metabolism*

Substances

  • Receptors, GABA-A
  • Flumazenil