K-opioid receptor changes in experimental models of cerebral ischaemia and atherosclerosis in the rabbit

Pharmacol Res. 1992 Dec;26(4):409-15. doi: 10.1016/1043-6618(92)90240-c.

Abstract

Thromboembolic phenomena and transient ischaemic attacks (TIA) are considered the basis of ischaemic pathologies. The aim of the present research is to investigate the involvement of k-opioid receptors in cerebral blood flow (CBF) impairment which results in experimental stroke or dietary atherosclerosis in rabbits. CBF measurement showed a significant decrease in rabbits submitted to embolization and/or atherosclerosis. Binding studies showed that massive cerebral ischaemia and atherosclerosis produced a significant increase in the number of k-opioid receptors (Bmax), without changing (KD) affinity values. In conclusion, the results obtained seem to indicate that the increase in k-opioid receptors might play a crucial role in a common cerebral biochemical mechanism both in ischaemic and atherosclerotic pathologies.

MeSH terms

  • Animals
  • Arteriosclerosis / metabolism*
  • Arteriosclerosis / physiopathology
  • Brain Ischemia / metabolism*
  • Brain Ischemia / physiopathology
  • Cerebral Cortex / drug effects
  • Cerebral Cortex / metabolism
  • Cerebrovascular Circulation / physiology
  • Diet, Atherogenic
  • Dynorphins / metabolism
  • Electroencephalography / drug effects
  • Evoked Potentials, Somatosensory / drug effects
  • Kinetics
  • Lipids / blood
  • Rabbits
  • Receptors, Opioid, kappa / metabolism*

Substances

  • Lipids
  • Receptors, Opioid, kappa
  • Dynorphins