Structure-activity relationships for unsaturated dialdehydes. 6. The mutagenic activity of 11 compounds in the V79/HGPRT assay

Mutat Res. 1992 Aug;268(2):315-21. doi: 10.1016/0027-5107(92)90237-v.

Abstract

The mutagenic activity of 11 sesquiterpenoid unsaturated dialdehydes in the V79/HGPRT assay has been determined, and is compared with previously published data on the mutagenicity of the same compounds towards Ames Salmonella strains. One compound, isovelleral, is a potent mutagen in both assays, while six compounds, which are positive in the Ames Salmonella/microsome assay, show no significant activity in this study. One compound, acetylmerulidial, is negative in the Ames Salmonella/microsome assay but significantly although weakly mutagenic in the V79/HGPRT assay. The remaining three compounds are inactive in both assays. The study is part of a general investigation of quantitative structure-activity relationships for unsaturated dialdehydes, a class of natural occurring compounds known for their potent and numerous biological activities.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aldehydes / chemistry*
  • Aldehydes / toxicity*
  • Animals
  • Cricetinae
  • Cricetulus
  • Genes
  • Hypoxanthine Phosphoribosyltransferase / genetics
  • Mutagenesis*
  • Mutagenicity Tests / methods
  • Mutagens / chemistry
  • Sesquiterpenes / chemistry*
  • Sesquiterpenes / toxicity*
  • Structure-Activity Relationship

Substances

  • Aldehydes
  • Mutagens
  • Sesquiterpenes
  • Hypoxanthine Phosphoribosyltransferase