Presence of the binding of a variety of ligands related to ionotropic excitatory amino acid receptors in rat retina

Brain Res. 1992 Mar 27;576(1):168-72. doi: 10.1016/0006-8993(92)90626-k.

Abstract

The binding of [3H]L-glutamic (Glu), [3H](+/-)-3-(2-carboxypiperazin-4-yl)propyl-1-phosphonic and [3H]D,L-(E)-2-amino-4-propyl-5-phosphono-3-pentenoic acids was detected in rat retinal membranes extensively washed and treated with a low concentration of Triton X-100, in addition to the binding of both [3H]glycine (Gly) and [3H]5,7-dichlorokynurenic acid. Furthermore, retinal membranes exhibited the binding of [3H](+)-5-methyl-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5,10-imi ne in the presence of Glu, Gly and spermidine irrespective of the incubation period employed. Rat retina also contained the binding of [3H]kainic acid as well as the binding of [3H]alpha-amino-3-hydroxy-5-methylisoxazole-4-propionic acid which was sensitive to potentiation by potassium thiocyanate. In addition, the binding of both [3H](+)-3-(hydroxyphenyl)-N-(l-propyl)piperidine and [3H]1,3-di-o-tolyl-guanidine was found in rat retinal membranes extensively washed but not treated with Triton X-100. These results give support for the proposal that the rodent retina contains subclasses of ionotropic brain excitatory amino acid receptors including the N-methyl-D-aspartate receptor ionophore complex as well as sigma sites.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Membrane / metabolism
  • Glycine / metabolism
  • Ibotenic Acid / analogs & derivatives
  • Ibotenic Acid / metabolism
  • Kinetics
  • Male
  • Radioligand Assay
  • Rats
  • Rats, Inbred Strains
  • Receptors, AMPA
  • Receptors, Glycine
  • Receptors, N-Methyl-D-Aspartate / metabolism*
  • Receptors, Neurotransmitter / metabolism*
  • Retina / metabolism*
  • Tritium
  • alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid

Substances

  • Receptors, AMPA
  • Receptors, Glycine
  • Receptors, N-Methyl-D-Aspartate
  • Receptors, Neurotransmitter
  • Tritium
  • Ibotenic Acid
  • alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid
  • Glycine