Helicobacter pylori stimulates host cyclooxygenase-2 gene transcription: critical importance of MEK/ERK-dependent activation of USF1/-2 and CREB transcription factors

Cell Microbiol. 2003 Nov;5(11):821-34. doi: 10.1046/j.1462-5822.2003.00324.x.

Abstract

Cyclooxygenase-2 (COX-2) represents the inducible key enzyme of arachidonic acid metabolism and contributes to the pathogenesis of gastroduodenal ulcers and gastric cancer. Helicobacter pylori infection is associated with elevated gastric COX-2 levels, but the mechanisms underlying H. pylori-dependent cox-2 gene expression are unclear. H. pylori stimulated cox-2 mRNA and protein abundance in gastric epithelial cells in vitro and in vivo, and functional analysis of the cox-2 gene promoter mapped its H. pylori-responsive region to a proximal CRE/Ebox element at -56 to -48. Moreover, USF1/-2 and CREB transcription factors binding to this site were identified to transmit H. pylori-dependent cox-2 transcription. Activation of MEK/ERK1/-2 signalling by bacterial virulence factors located outside the H. pylori cag pathogenicity island (cagPAI) was found to mediate bacterial effects on the cox-2 promoter. Our study provides a detailed description of the molecular pathways underlying H. pylori-dependent cox-2 gene expression in gastric epithelial cells, and may thus contribute to a better understanding of mechanisms underlying H. pylori pathogenicity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cyclic AMP Response Element-Binding Protein / metabolism*
  • Cyclooxygenase 2
  • DNA-Binding Proteins*
  • Epithelial Cells / metabolism
  • Gastric Mucosa / cytology
  • Gastric Mucosa / metabolism
  • Gene Expression Regulation
  • Helicobacter Infections / microbiology*
  • Helicobacter pylori / genetics
  • Helicobacter pylori / metabolism*
  • Isoenzymes / genetics*
  • Isoenzymes / metabolism
  • MAP Kinase Kinase Kinases / metabolism*
  • MAP Kinase Signaling System / physiology
  • Mice
  • Mitogen-Activated Protein Kinases / metabolism*
  • Promoter Regions, Genetic
  • Prostaglandin-Endoperoxide Synthases / genetics*
  • Prostaglandin-Endoperoxide Synthases / metabolism
  • Transcription Factors / metabolism*
  • Transcription, Genetic
  • Upstream Stimulatory Factors
  • Virulence Factors / genetics
  • Virulence Factors / metabolism

Substances

  • Cyclic AMP Response Element-Binding Protein
  • DNA-Binding Proteins
  • Isoenzymes
  • Transcription Factors
  • Upstream Stimulatory Factors
  • Usf1 protein, mouse
  • Virulence Factors
  • Cyclooxygenase 2
  • Prostaglandin-Endoperoxide Synthases
  • Mitogen-Activated Protein Kinases
  • MAP Kinase Kinase Kinases