[The prolonged use of calcium antagonists in myocardial infarct in rats: their effect on hemodynamics and the contractile function and morphology of the heart muscle]

Eksp Klin Farmakol. 1992 May-Jun;55(3):17-20.
[Article in Russian]

Abstract

Experiments on rats with myocardial infarction induced by occlusion of the left coronary artery were made to explore the influence of calcium antagonists injected intraperitoneally for a long time (daily, for 21 days) on hemodynamics, contractile function and morphology of the heart muscle. It has been shown that verapamil (0.5 mg/kg), diltiazem (2 mg/kg) and nimodipine (20 micrograms/kg) do not exert under those conditions any noticeable effect on pump and contractile heart functions. Administration of verapamil in a doze of 2 mg/kg enhanced heart failure. The drugs under study normalized the response of contractile heart function to volumetric load, which is related to a considerable measure to the acceleration of reparative processes in the myocardium.

Publication types

  • Comparative Study
  • English Abstract

MeSH terms

  • Animals
  • Calcium Channel Blockers / pharmacology
  • Calcium Channel Blockers / therapeutic use*
  • Diltiazem / pharmacology
  • Diltiazem / therapeutic use
  • Drug Evaluation, Preclinical
  • Heart / drug effects*
  • Heart / physiopathology
  • Hemodynamics / drug effects
  • Male
  • Myocardial Contraction / drug effects*
  • Myocardial Infarction / drug therapy*
  • Myocardial Infarction / physiopathology
  • Myocardium / pathology*
  • Nimodipine / pharmacology
  • Nimodipine / therapeutic use
  • Rats
  • Time Factors
  • Verapamil / pharmacology
  • Verapamil / therapeutic use

Substances

  • Calcium Channel Blockers
  • Nimodipine
  • Verapamil
  • Diltiazem