Novel nanosensors for rapid analysis of telomerase activity

Cancer Res. 2004 Jan 15;64(2):639-43. doi: 10.1158/0008-5472.can-03-2798.

Abstract

Elevated telomerase levels are found in many malignancies, offering an attractive target for therapeutic intervention and diagnostic or prognostic purposes. Here we describe the use of a novel nanosensor developed for rapid screens of telomerase activity in biological samples. The technique utilizes magnetic nanoparticles that, on annealing with telomerase synthesized TTAGGG repeats, switch their magnet state, a phenomenon readily detectable by magnetic readers. We tested the efficacy of different telomerase inhibitors in crude human and murine samples and show that phosphorylation of telomerase regulates its activity. High-throughput adaptation of the technique by magnetic resonance imaging allowed processing of hundreds of samples within tens of minutes at ultrahigh sensitivities. Together, these studies establish and validate a novel and powerful tool for rapidly sensing telomerase activity and provide the rationale for developing analogous magnetic nanoparticles for in vivo sensing.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Biosensing Techniques
  • Cell Line
  • Cell Line, Tumor
  • Female
  • Humans
  • Kinetics
  • Male
  • Microscopy, Atomic Force / methods
  • Oligodeoxyribonucleotides / chemistry
  • Oligodeoxyribonucleotides / metabolism
  • Sensitivity and Specificity
  • Telomerase / analysis*
  • Telomerase / antagonists & inhibitors
  • Telomerase / metabolism

Substances

  • Oligodeoxyribonucleotides
  • Telomerase