Involvement of rho-kinase pathway in contractile activity of rabbit RPE cells in vivo and in vitro

Invest Ophthalmol Vis Sci. 2004 Feb;45(2):668-74. doi: 10.1167/iovs.02-0808.

Abstract

Purpose: Increased alpha-smooth muscle actin (alpha-SMA) expression in epiretinal membranes causes tractional retinal detachment (TRD) in proliferative vitreoretinopathy (PVR). The Rho-A/Rho-associated kinase signaling pathway is a principal mediator of contractile force generation in nonmuscle cells. In the current study, the relation between the Rho-kinase pathway and alpha-SMA expression and type I collagen gel contractile activity in retinal pigment epithelial (RPE) cells was investigated, using Y27632, a specific inhibitor of p160ROCK, and the involvement of the Rho-kinase pathway was evaluated in a rabbit PVR model with cultured RPE cells and platelet-rich plasma (PRP).

Methods: RPE cells were obtained from rabbits and cultured. The number of passages and the effect of Y27632 on alpha-SMA expression were studied by immunohistochemistry and immunoblot analysis. An in vitro type I collagen gel contraction assay and MTT assay evaluated the effect of Y27632 on RPE cell contractile force and proliferation. Cultured sixth-passage rabbit RPE cells were coinjected with PRP intravitreally, followed by 50 micro M of Y27632, injected weekly. The presence of TRD was assessed until 28 days to evaluate the effect of Y27632 in vivo.

Results: Expression of alpha-SMA was increased according to the passages. Y27632 suppressed alpha-SMA expression in cultured RPE cells and impaired contractile force. Y27632 did not affect the proliferative potential. Y27632 significantly (P < 0.01) reduced TRD development.

Conclusions: Y27632 decreased alpha-SMA expression and the contractile force generated by RPE cells and attenuated PVR, indicating the involvement of the Rho-kinase pathway in cell-dependent collagen contraction in vitro and in vivo. The drug may affect the biological event by inhibiting alpha-SMA expression, and Y27632 could be useful for preventing PVR.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Actins / metabolism*
  • Amides / pharmacology*
  • Animals
  • Cell Division / drug effects
  • Cells, Cultured
  • Collagen Type I / metabolism*
  • Enzyme Inhibitors / pharmacology*
  • Female
  • Immunoblotting
  • Immunohistochemistry
  • Intracellular Signaling Peptides and Proteins
  • Male
  • Pigment Epithelium of Eye / cytology
  • Pigment Epithelium of Eye / enzymology*
  • Protein Serine-Threonine Kinases / antagonists & inhibitors
  • Protein Serine-Threonine Kinases / physiology*
  • Pyridines / pharmacology*
  • Rabbits
  • Vitreoretinopathy, Proliferative / enzymology
  • Vitreoretinopathy, Proliferative / prevention & control
  • rho-Associated Kinases

Substances

  • Actins
  • Amides
  • Collagen Type I
  • Enzyme Inhibitors
  • Intracellular Signaling Peptides and Proteins
  • Pyridines
  • Y 27632
  • Protein Serine-Threonine Kinases
  • rho-Associated Kinases