Characterization of a single-chain intrabody directed against the human receptor tyrosine kinase Ron

J Immunol Methods. 2004 Feb 1;285(1):99-109. doi: 10.1016/j.jim.2003.11.003.

Abstract

A large human nonimmune phage antibody library was screened by affinity chromatography to select single-chain antibodies directed against the human receptor tyrosine kinase (RTK) Ron. As antigen, we used a GST fusion protein (GST-IRP(-)) containing the whole intracellular portion of Ron except for the carboxyl-terminal arginine-proline-rich motif. One selected phage was highly specific for Ron when tested in an enzyme-linked immunosorbent assay (ELISA). We report here the immunological characterization of this anti-Ron single-chain antibody (sc7) and show that it recognizes both denatured and native forms of the receptor. The epitope bound by sc7 maps within the first 50 amino acid residues of the juxtamembrane domain of Ron. This monoclonal fragment does not cross-react with other receptor tyrosine kinases including the closely related human proto-oncogene Met. We demonstrate that the isolated antibody fragment interacts in vivo with the intracellular domain of Ron in mammalian cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antibodies / genetics*
  • Antibody Specificity
  • Antigen-Antibody Reactions
  • Base Sequence
  • Cell Line
  • Chromatography, Affinity
  • Cross Reactions
  • Dogs
  • Enzyme-Linked Immunosorbent Assay
  • Epitope Mapping
  • Epitopes / genetics
  • Humans
  • Immunoglobulin Variable Region / genetics
  • Peptide Library
  • Plasmids / genetics
  • Precipitin Tests
  • Proto-Oncogene Mas
  • Receptor Protein-Tyrosine Kinases / genetics
  • Receptor Protein-Tyrosine Kinases / immunology*
  • Receptor Protein-Tyrosine Kinases / isolation & purification
  • Recombinant Fusion Proteins / genetics
  • Recombinant Fusion Proteins / immunology

Substances

  • Antibodies
  • Epitopes
  • Immunoglobulin Variable Region
  • MAS1 protein, human
  • Peptide Library
  • Proto-Oncogene Mas
  • Recombinant Fusion Proteins
  • RON protein
  • Receptor Protein-Tyrosine Kinases