Primary antibody response to keyhole limpet hemocyanin in rat as a model for immunotoxicity evaluation

Toxicology. 2004 Apr 1;197(1):23-35. doi: 10.1016/j.tox.2003.12.003.

Abstract

To address current regulatory expectations on immunotoxicity testing of new chemicals, we describe an animal model that measures the primary antibody response to the T-cell dependent antigen, keyhole limpet hemocyanin (KLH). Single immunization with KLH by either footpad (300microg/rat) or intravenous (300microg/kg) route in Sprague Dawley rats resulted in increased germinal center formation in the spleen and a robust anti-KLH IgM (70-388microg/ml) and IgG (230-470microg/ml) antibody response with peak detection on Days 5 and 14 post-immunization, respectively. Subcutaneous immunization with KLH (300microg/kg) resulted in a much weaker anti-KLH IgM and IgG (< or =20microg/ml) antibody response with no detectable increase in splenic germinal center formation. The utility of a rat KLH immunization model in detecting immunosuppression was evaluated with the known immunosuppressive drugs: cyclosporin, azathioprine and prednisolone. Rats, treated with drug at a maximum tolerated dose, were immunized with KLH by footpad or intravenous injection and serum samples were collected at various intervals up to 2 weeks post-immunization. Additional study parameters included terminal body weight, hematology and/or histopathology. All three drugs inhibited the IgM (60%) and IgG (> or =90%) antibody responses in the absence of overt toxicity based on evaluation of the standard toxicology parameters. In conclusion, measurement of a rat primary antibody response to KLH by ELISA is a reliable and readily standardized method for assessing immunotoxicity of pharmaceuticals.

MeSH terms

  • Animals
  • Antibody Formation / drug effects*
  • Antibody Formation / immunology
  • Antigens / administration & dosage
  • Antigens / pharmacology*
  • Enzyme-Linked Immunosorbent Assay
  • Female
  • Foot
  • Hemocyanins / administration & dosage
  • Hemocyanins / immunology
  • Hemocyanins / pharmacology*
  • Hindlimb
  • Hyperplasia / etiology
  • Hyperplasia / pathology
  • Immunity, Cellular / drug effects*
  • Immunity, Cellular / immunology
  • Immunocompromised Host
  • Immunoglobulin G / analysis
  • Immunoglobulin G / biosynthesis
  • Immunoglobulin M / analysis
  • Immunoglobulin M / biosynthesis
  • Immunosuppression Therapy / adverse effects
  • Immunosuppressive Agents / classification
  • Immunosuppressive Agents / toxicity*
  • Injections
  • Male
  • Models, Animal
  • Pulmonary Alveoli / pathology
  • Rats
  • Rats, Sprague-Dawley
  • Respiratory Tract Infections / immunology
  • Respiratory Tract Infections / pathology

Substances

  • Antigens
  • Immunoglobulin G
  • Immunoglobulin M
  • Immunosuppressive Agents
  • Hemocyanins
  • keyhole-limpet hemocyanin