NMDA receptor alterations in neurons from pediatric cortical dysplasia tissue

Cereb Cortex. 2004 Jun;14(6):634-46. doi: 10.1093/cercor/bhh024. Epub 2004 Mar 28.

Abstract

The subunit composition of glutamate receptors affects their functional properties, and could contribute to abnormal electrophysiology in pediatric cortical dysplasia (CD). We examined electrophysiological responses and subunit assembly of N-methyl-D-aspartate (NMDA) receptors in acutely dissociated normal-appearing pyramidal and cytomegalic neurons from CD tissue and normal-appearing pyramidal neurons from non-CD tissue. In most cytomegalic and approximately 30% of normal-appearing pyramidal neurons from CD tissue, NMDA currents showed decreased Mg(2+) sensitivity compared with neurons from non-CD tissue. Ifenprodil had less effect in CD compared with non-CD neurons, indicating a functional loss of NR2B subunits. NMDA-evoked current density was decreased in cytomegalic compared with normal-appearing neurons. Single-cell reverse transcriptase polymerase chain reaction showed that all non-CD neurons expressed NR2B subunit mRNA. By comparison, 22% of pyramidal neurons in CD tissue lacked NR2B mRNA. Immunofluorescence showed a decrease in NR2B subunit expression in cytomegalic neurons and a subset of normal-appearing pyramidal neurons from CD tissue. Taken together, these results demonstrate the presence of NMDA receptors with altered subunit composition and Mg(2+) sensitivity that could contribute to functional abnormalities in CD.

Publication types

  • Clinical Trial
  • Comparative Study
  • Controlled Clinical Trial
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adolescent
  • Cells, Cultured
  • Cerebral Cortex / abnormalities*
  • Cerebral Cortex / drug effects
  • Cerebral Cortex / physiopathology*
  • Child
  • Child, Preschool
  • Epilepsy / pathology*
  • Epilepsy / physiopathology*
  • Humans
  • Infant
  • Magnesium / pharmacology
  • Membrane Potentials / drug effects
  • N-Methylaspartate / pharmacology
  • Piperidines / pharmacology
  • Pyramidal Cells / drug effects
  • Pyramidal Cells / metabolism*
  • Pyramidal Cells / physiopathology*
  • Receptors, N-Methyl-D-Aspartate / chemistry
  • Receptors, N-Methyl-D-Aspartate / drug effects
  • Receptors, N-Methyl-D-Aspartate / metabolism*
  • Reference Values

Substances

  • Piperidines
  • Receptors, N-Methyl-D-Aspartate
  • N-Methylaspartate
  • Magnesium
  • ifenprodil