Effect of donepezil on group II mGlu receptor agonist- or antagonist-induced amnesia on passive avoidance in mice

Neural Plast. 2003;10(4):319-25. doi: 10.1155/NP.2003.319.

Abstract

We examined the effect of the acetylcholinesterase (AChE) inhibitor, donepezil hydrocloride (DONP), on group II metabotropic glutamate (mGlu) receptor agonist- or antagonist-induced amnesia in the step-through passive avoidance task in male mice. DCG-IV, a group II mGlu receptor agonist, at dose of 50 ng and LY341495, a group II mGlu receptor antagonist, at dose of 300 ng, significantly attenuated the latency on the step-through task. The subcutaneous injection of DONP at dose of 1 mg/kg 1 hour before passive avoidance performance ameliorated the amnesia induced by DCG-IV and LY341495, whereas donepezil alone did not affect task latency. The results suggest that activation of group II mGlu receptors and disinhibition of the cAMP/PKA signaling pathway (caused by group II mGlu receptor antagonist) have a negative action on step-through passive avoidance memory performance, and that group II mGlu receptors and ACh interact to modulate learning and memory function.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acids / pharmacology
  • Amnesia / chemically induced*
  • Amnesia / prevention & control*
  • Animals
  • Avoidance Learning / drug effects*
  • Cholinesterase Inhibitors / pharmacology*
  • Cyclopropanes / pharmacology
  • Donepezil
  • Excitatory Amino Acid Antagonists / pharmacology
  • Glycine / analogs & derivatives*
  • Glycine / pharmacology
  • Indans / pharmacology*
  • Male
  • Memory / drug effects
  • Mice
  • Nootropic Agents / pharmacology*
  • Piperidines / pharmacology*
  • Receptors, Metabotropic Glutamate / agonists*
  • Receptors, Metabotropic Glutamate / antagonists & inhibitors*
  • Xanthenes / pharmacology

Substances

  • Amino Acids
  • Cholinesterase Inhibitors
  • Cyclopropanes
  • Excitatory Amino Acid Antagonists
  • Indans
  • LY 341495
  • Nootropic Agents
  • Piperidines
  • Receptors, Metabotropic Glutamate
  • Xanthenes
  • metabotropic glutamate receptor 2
  • 2-(2,3-dicarboxycyclopropyl)glycine
  • Donepezil
  • Glycine