Dose dependence of N-hydroxy-3,2'-dimethyl-4-aminobiphenyl-induced rat prostate carcinogenesis

Jpn J Cancer Res. 1992 Jul;83(7):695-8. doi: 10.1111/j.1349-7006.1992.tb01968.x.

Abstract

Groups of F344 rats were administered biweekly intraperitoneal injections of N-hydroxy-3,2'-dimethyl-4-aminobiphenyl (N-OH-DMAB) at a dose of 5, 10 or 20 mg/kg body weight or DMAB, the parent compound, at a dose of 25 mg/kg body weight, for a total of 10 times. Prostate carcinomas in the ventral lobe developed in a N-OH-DMAB dose-dependent manner (0, 17.6 and 66.7%, respectively) with limited tumor yields in other organs. Although intraperitoneal administration of DMAB was similarly found to induce prostate tumors, it also caused severe chemical peritonitis, which resulted in a high mortality. The present data confirmed that intraperitoneal administration of N-OH-DMAB provides a relatively specific induction method for models of prostate carcinogenesis.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aminobiphenyl Compounds*
  • Animals
  • Carcinogens*
  • Disease Models, Animal
  • Dose-Response Relationship, Drug
  • Injections, Intraperitoneal
  • Male
  • Prostatic Neoplasms / chemically induced*
  • Rats
  • Rats, Inbred F344

Substances

  • Aminobiphenyl Compounds
  • Carcinogens
  • 2',3-dimethyl-4-aminobiphenyl
  • N-hydroxy-3,2'-dimethyl-4-aminobiphenyl