Long-term pharmacokinetics of amprenavir in combination with delavirdine in HIV-infected children

AIDS. 2004 Jul 2;18(10):1473-5. doi: 10.1097/01.aids.0000131342.53419.4d.

Abstract

Five heavily pretreated HIV-infected children were put on amprenavir and delavirdine plus two nucleoside inhibitors to reverse transcriptase to boost amprenavir levels and to use the antiretroviral activity of a non-nucleoside reverse transcriptase inhibitor. No data are available about this combination in children. It w;as well tolerated, and the median reduction in viral load was 1.5 log after 18 months. Delavirdine boosted amprenavir trough levels more than 10-fold, and delavirdine trough levels remained i several fold above susceptible HIV strains.

MeSH terms

  • Adolescent
  • Anti-HIV Agents / pharmacokinetics*
  • Area Under Curve
  • Carbamates
  • Child
  • Delavirdine / pharmacokinetics*
  • Drug Combinations
  • Furans
  • HIV Infections / drug therapy*
  • Humans
  • Reverse Transcriptase Inhibitors / pharmacokinetics*
  • Sulfonamides / pharmacokinetics*

Substances

  • Anti-HIV Agents
  • Carbamates
  • Drug Combinations
  • Furans
  • Reverse Transcriptase Inhibitors
  • Sulfonamides
  • amprenavir
  • Delavirdine