Structure of the N-terminal half of gelsolin bound to actin: roles in severing, apoptosis and FAF

EMBO J. 2004 Jul 21;23(14):2713-22. doi: 10.1038/sj.emboj.7600280. Epub 2004 Jun 24.

Abstract

The actin filament-severing functionality of gelsolin resides in its N-terminal three domains (G1-G3). We have determined the structure of this fragment in complex with an actin monomer. The structure reveals the dramatic domain rearrangements that activate G1-G3, which include the replacement of interdomain interactions observed in the inactive, calcium-free protein by new contacts to actin, and by a novel G2-G3 interface. Together, these conformational changes are critical for actin filament severing, and we suggest that their absence leads to the disease Finnish-type familial amyloidosis. Furthermore, we propose that association with actin drives the calcium-independent activation of isolated G1-G3 during apoptosis, and that a similar mechanism operates to activate native gelsolin at micromolar levels of calcium. This is the first structure of a filament-binding protein bound to actin and it sets stringent, high-resolution limitations on the arrangement of actin protomers within the filament.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Actins / chemistry
  • Actins / metabolism*
  • Amyloidosis, Familial / metabolism*
  • Animals
  • Apoptosis*
  • Binding Sites
  • Calcium / metabolism
  • Crystallography, X-Ray
  • Gelsolin / chemistry*
  • Gelsolin / genetics
  • Gelsolin / isolation & purification
  • Gelsolin / metabolism*
  • Horses
  • Humans
  • Models, Molecular
  • Mutation
  • Protein Binding
  • Protein Conformation
  • Protein Structure, Secondary
  • Protein Structure, Tertiary
  • Structure-Activity Relationship

Substances

  • Actins
  • Gelsolin
  • Calcium

Associated data

  • PDB/1RGI