Effects of co-administration of ibuprofen-lysine on the pharmacokinetics of amikacin in preterm infants during the first days of life

Biol Neonate. 2004;86(3):207-11. doi: 10.1159/000079618. Epub 2004 Jul 7.

Abstract

The aim of this study was to assess the effects of intravenous co-administration of ibuprofen-lysine on the pharmacokinetics of amikacin during the first days of life in preterm infants. The pharmacokinetics of amikacin were retrospectively calculated in a cohort of 73 neonates (gestational age <31 weeks) who received either ibuprofen-lysine or placebo following inclusion in the multicentre ibuprofen prophylaxis study. Assuming a one-compartment model with instantaneous input and first-order output, there was no significant difference in the median distribution volume (0.63 vs. 0.59 liters/kg), but the median serum half-life (16.4 vs. 12.4 h) of amikacin was significantly longer (p <0.02), and the clearance (0.36 vs. 0.6 ml/kg/min; p <0.005) of amikacin was significantly lower in infants who received ibuprofen-lysine. We conclude that the time interval between consecutive amikacin administrations should be prolonged, if ibuprofen-lysine is co-administered.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amikacin / pharmacokinetics*
  • Bacterial Infections / prevention & control
  • Double-Blind Method
  • Gestational Age
  • Half-Life
  • Humans
  • Ibuprofen / administration & dosage*
  • Infant, Newborn
  • Infant, Premature*
  • Infant, Premature, Diseases / prevention & control
  • Infusions, Intravenous
  • Lysine / administration & dosage*
  • Metabolic Clearance Rate
  • Placebos
  • Retrospective Studies

Substances

  • Placebos
  • Amikacin
  • Lysine
  • Ibuprofen