Vav2 as a Rac-GDP/GTP exchange factor responsible for the nectin-induced, c-Src- and Cdc42-mediated activation of Rac

J Biol Chem. 2005 Feb 11;280(6):4940-7. doi: 10.1074/jbc.M408710200. Epub 2004 Oct 13.

Abstract

Nectins are Ca2+-independent immunoglobulin-like cell-cell adhesion molecules that form homo- and hetero-trans-dimers (trans-interactions). Nectins first form cell-cell contact and then recruit cadherins to the nectin-based cell-cell contact sites to form adherens junctions cooperatively with cadherins. In addition, the trans-interactions of nectins induce the activation of Cdc42 and Rac small G proteins, which enhances the formation of adherens junctions by forming filopodia and lamellipodia, respectively. The trans-interactions of nectins first recruit and activate c-Src at the nectin-based cell-cell contact sites. c-Src then phosphorylates and activates FRG, a Cdc42-GDP/GTP exchange factor (GEF) for Cdc42. The activation of both c-Src and Cdc42 by FRG is necessary for the activation of Rac, but the Rac-GEF responsible for this activation of Rac remains unknown. We showed here that the nectin-induced activation of Rac was inhibited by a dominant negative mutant of Vav2, a Rac-GEF. Nectins recruited and tyrosine-phosphorylated Vav2 through c-Src at the nectin-based cell-cell contact sites, whereas Cdc42 was not necessary for the nectin-induced recruitment of Vav2 or the nectin-induced, c-Src-mediated tyrosine phosphorylation of Vav2. Cdc42 activated through c-Src then enhanced the GEF activity of tyrosine-phosphorylated Vav2 on Rac1. These results indicate that Vav2 is a GEF responsible for the nectin-induced, c-Src-, and Cdc42-mediated activation of Rac.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • CSK Tyrosine-Protein Kinase
  • Calcium / metabolism
  • Cell Adhesion
  • Cell Adhesion Molecules / chemistry
  • Cell Adhesion Molecules / metabolism*
  • Cell Line
  • Dogs
  • Fibroblasts / metabolism
  • Genes, Dominant
  • Guanine Nucleotide Exchange Factors / physiology*
  • Immunoprecipitation
  • Mice
  • Microscopy, Fluorescence
  • Models, Biological
  • Mutation
  • Nectins
  • Oncogene Proteins / metabolism
  • Oncogene Proteins / physiology*
  • Phosphorylation
  • Plasmids / metabolism
  • Protein Binding
  • Protein Structure, Tertiary
  • Protein-Tyrosine Kinases / metabolism*
  • Proto-Oncogene Proteins c-vav
  • Pseudopodia / metabolism
  • Time Factors
  • Transfection
  • Transgenes
  • Tyrosine / chemistry
  • Tyrosine / metabolism
  • cdc42 GTP-Binding Protein / metabolism*
  • rac GTP-Binding Proteins / metabolism*
  • src-Family Kinases

Substances

  • Cell Adhesion Molecules
  • Guanine Nucleotide Exchange Factors
  • Nectins
  • Oncogene Proteins
  • Proto-Oncogene Proteins c-vav
  • Vav2 protein, mouse
  • Tyrosine
  • Protein-Tyrosine Kinases
  • CSK Tyrosine-Protein Kinase
  • src-Family Kinases
  • cdc42 GTP-Binding Protein
  • rac GTP-Binding Proteins
  • Calcium