Role of manidipine in the management of patients with hypertension

Expert Rev Cardiovasc Ther. 2004 Nov;2(6):815-27. doi: 10.1586/14779072.2.6.815.

Abstract

Manidipine is a third-generation dihydropyridine calcium antagonist, which causes systemic vasodilation by inhibiting the voltage-dependent calcium inward currents in smooth muscle cells. In clinical studies, manidipine has been shown to significantly lower office and 24-h blood pressure compared with placebo in patients with essential hypertension. The resulting reduction in blood pressure is maintained over 24 h, with preservation of the circadian blood pressure pattern; its blood pressure-lowering capacity appears to be similar to that of other calcium antagonists. In elderly patients with mild-to-moderate essential hypertension, manidipine is able to significantly decrease blood pressure compared with placebo for up to 3 years of treatment. The drug also significantly lowers blood pressure in patients with hypertension and concomitant Type 2 diabetes mellitus or renal impairment, and is devoid of adverse metabolic effects. It is well-tolerated with few untoward adverse effects related to vasodilation. In particular, manidipine appears to have less potential for pedal edema than other calcium channel blockers.

Publication types

  • Comparative Study

MeSH terms

  • Adult
  • Aged
  • Animals
  • Biological Availability
  • Blood Pressure Monitoring, Ambulatory
  • Dihydropyridines / administration & dosage*
  • Dihydropyridines / pharmacokinetics*
  • Disease Models, Animal
  • Dose-Response Relationship, Drug
  • Drug Administration Schedule
  • Female
  • Follow-Up Studies
  • Humans
  • Hypertension / diagnosis
  • Hypertension / drug therapy*
  • Male
  • Maximum Tolerated Dose
  • Middle Aged
  • Nitrobenzenes
  • Piperazines
  • Randomized Controlled Trials as Topic
  • Risk Assessment
  • Severity of Illness Index
  • Treatment Outcome

Substances

  • Dihydropyridines
  • Nitrobenzenes
  • Piperazines
  • manidipine