Comparison of the effect of amphotericin B desoxycholate and amphotericin B colloidal dispersion on renal functions and renal morphology in rats

Nephrology (Carlton). 2005 Feb;10(1):57-62. doi: 10.1111/j.1440-1797.2005.00339.x.

Abstract

Background and aim: Amphotericin B (AmB) desoxycholate remains as one of the most efficacious agents currently available for the treatment of systemic fungal infections; however, amphotericin B colloidal dispersion (ABCD) has been developed because of AmB desoxycholate nephrotoxicity. The goal of our study was to compare the effect of administration of AmB desoxycholate and ABCD on renal functions and renal morphology in rats.

Results: Amophotericin B desoxycholate as well as ABCD causes damage to renal tubuli and polyuria. Amophotericin desoxycholate causes considerably more severe damage to tubuli than ABCD, but the morphological damage to renal glomeruli is minimal in both formulas. In tubular cells, AmB desoxycholate causes severe damage to mitochondria, vacuolation of cytoplasm, and increased values of volume density of peroxisomes.

Conclusion: None of these formulas causes a decrease in glomerular filtration in rats when animals are properly hydrated.

Publication types

  • Comparative Study

MeSH terms

  • Amphotericin B / toxicity*
  • Animals
  • Antifungal Agents / toxicity*
  • Cytoplasm / drug effects
  • Cytoplasm / pathology
  • Deoxycholic Acid / toxicity*
  • Drug Combinations
  • Glomerular Filtration Rate / drug effects
  • Kidney Tubules, Collecting / drug effects
  • Kidney Tubules, Collecting / pathology
  • Kidney Tubules, Collecting / physiology
  • Kidney Tubules, Proximal / drug effects*
  • Kidney Tubules, Proximal / pathology
  • Kidney Tubules, Proximal / physiology*
  • Loop of Henle / drug effects
  • Loop of Henle / pathology
  • Loop of Henle / physiology
  • Male
  • Mitochondria / drug effects
  • Mitochondria / pathology
  • Models, Animal
  • Rats
  • Rats, Wistar
  • Vacuoles / drug effects
  • Vacuoles / pathology

Substances

  • Antifungal Agents
  • Drug Combinations
  • Deoxycholic Acid
  • Amphotericin B
  • amphotericin B, deoxycholate drug combination