Studies on the apoptotic activity of natural and synthetic retinoids: discovery of a new class of synthetic terphenyls that potently support cell growth and inhibit apoptosis in neuronal and HL-60 cells

J Med Chem. 2005 Jun 30;48(13):4293-9. doi: 10.1021/jm049080y.

Abstract

New terphenyl derivatives have been synthesized and tested for their effect on cell survival in serum-free cultures. These compounds protected HL60 cells from death and supported their growth with an activity higher than that of the natural 14-hydroxy-retro-retinol. Terphenyls 26 and 28 also possess antiapoptotic activity on neuronal cells, proving them as possible candidates for the treatment of neurodegenerative and ischemic diseases.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Apoptosis / drug effects*
  • Cell Division / drug effects
  • HL-60 Cells
  • Humans
  • Indicators and Reagents
  • Neurons / cytology
  • Neurons / drug effects
  • Neurons / physiology*
  • Retinoids / chemical synthesis*
  • Retinoids / chemistry
  • Retinoids / pharmacology*

Substances

  • Indicators and Reagents
  • Retinoids