Efficacy and safety of an oral formulation of cetirizine and prolonged-release pseudoephedrine versus budesonide nasal spray in the management of nasal congestion in allergic rhinitis

Treat Respir Med. 2005;4(4):283-7. doi: 10.2165/00151829-200504040-00006.

Abstract

Introduction: The aim of this study was to compare the decongestant properties and tolerability of oral cetirizine and pseudoephedrine in a prolonged release form with those of nasal (aqueous spray) budesonide.

Methods: Thirty-six individuals experiencing allergic rhinitis to house dustmites (HDM) participated in a study according to a randomized, crossover, two-period, two-treatment design with at least a 2-week washout period between treatments. In each period of 4 consecutive days, medications were taken twice daily. On day 1, immediately after the first intake of medication, individuals were exposed to HDM extract in the Vienna Challenge Chamber (VCC) for 5 hours. The primary efficacy parameter was nasal congestion, assessed by active anterior rhinomanometry and rating of nasal cavity photos.

Results: Rhinomanometry and nasal cavity photos both indicated that cetirizine/pseudoephedrine efficacy was statistically superior to budesonide in the management of nasal congestion during VCC sessions. The efficacy of cetirizine/pseudoephedrine was similar to that of budesonide from the end of day 1 up to day 4 when individuals were exposed to their natural environment post exposure to the aeroallergens. This study confirms the efficacy of cetirizine/pseudoephedrine and budesonide in the management of nasal congestion associated with allergic rhinitis. Both medications were well-tolerated. Cetirizine/pseudoephedrine was more effective than budesonide during HDM exposure, whereas budesonide became as effective as cetirizine/pseudoephedrine several hours post exposure to the allergens.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Intranasal
  • Administration, Oral
  • Adult
  • Anti-Allergic Agents / administration & dosage*
  • Budesonide / administration & dosage*
  • Cetirizine / administration & dosage*
  • Cross-Over Studies
  • Delayed-Action Preparations
  • Drug Combinations
  • Ephedrine / administration & dosage*
  • Female
  • Histamine H1 Antagonists, Non-Sedating / administration & dosage*
  • Humans
  • Male
  • Nasal Decongestants / administration & dosage*
  • Pulmonary Ventilation
  • Rhinitis, Allergic, Perennial / drug therapy*
  • Rhinitis, Allergic, Perennial / physiopathology
  • Rhinomanometry

Substances

  • Anti-Allergic Agents
  • Delayed-Action Preparations
  • Drug Combinations
  • Histamine H1 Antagonists, Non-Sedating
  • Nasal Decongestants
  • Budesonide
  • Ephedrine
  • Cetirizine