Lys-34, dispensable for integrase catalysis, is required for preintegration complex function and human immunodeficiency virus type 1 replication

J Virol. 2005 Oct;79(19):12584-91. doi: 10.1128/JVI.79.19.12584-12591.2005.

Abstract

Retroviral integrases (INs) function in the context of preintegration complexes (PICs). Two conserved Lys residues in the N-terminal domain of human immunodeficiency virus type 1 (HIV-1) IN were analyzed here for their roles in integration and virus replication. Whereas HIV-1(K46A) grew like the wild type, HIV-1(K34A) was dead. Yet recombinant IN(K34A) protein functioned in in vitro integration assays, and Vpr-IN(K34A) efficiently transcomplemented the infectivity defect of an IN active site mutant virus in cells. HIV-1(K34A) was therefore similar to a number of previously characterized mutant viruses that failed to replicate despite encoding catalytically competent IN. To directly analyze mutant PIC function, a sensitive PCR-based integration assay was developed. HIV-1(K34A) and related mutants failed to support detectable levels (<1% of wild type) of integration. We therefore concluded that mutations like K34A disrupted higher-order interactions important for PIC function/maturation compared to the innate catalytic activity of IN enzyme.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Substitution
  • HIV Integrase / chemistry
  • HIV Integrase / genetics*
  • HIV Integrase / physiology*
  • HIV-1 / genetics*
  • HIV-1 / physiology*
  • Mucoproteins / genetics
  • Mucoproteins / physiology*
  • Mutation, Missense
  • Polymerase Chain Reaction
  • Reverse Transcription
  • Virus Replication*

Substances

  • Mucoproteins
  • lysin, gastropoda
  • HIV Integrase