Role of HIV-1 minority populations on resistance mutational pattern evolution and susceptibility to protease inhibitors

AIDS. 2006 Jan 9;20(2):287-9. doi: 10.1097/01.aids.0000202650.03279.69.

Abstract

We investigated, in the protease and GAG cleavage sites, the role of minority populations on the evolution of resistance to a subsequent boosted protease inhibitor (PI) regimen after a first failure to nelfinavir. Two pathways were observed: the addition of mutations to a currently dominant genotype when minority variants are not shown, or the emergence of a minority variant as a dominant strain. These minor species, not detected by standard genotype, may influence PI susceptibility.

MeSH terms

  • Drug Resistance, Multiple, Viral / genetics*
  • Evolution, Molecular
  • Gene Products, gag / genetics
  • Genotype
  • HIV Infections / drug therapy*
  • HIV Infections / virology
  • HIV Protease / genetics
  • HIV Protease Inhibitors / therapeutic use*
  • HIV-1 / classification
  • HIV-1 / drug effects*
  • HIV-1 / genetics
  • Humans
  • Nelfinavir / therapeutic use
  • Treatment Failure

Substances

  • Gene Products, gag
  • HIV Protease Inhibitors
  • HIV Protease
  • Nelfinavir