Blockade of the interaction of leukotriene b4 with its receptor prevents development of autoimmune uveitis

Invest Ophthalmol Vis Sci. 2006 Apr;47(4):1543-9. doi: 10.1167/iovs.05-1238.

Abstract

Purpose: To investigate the role of leukotriene B4 (LTB4) and its receptor BLT1 in the pathogenesis of mouse uveitis.

Methods: Experimental autoimmune uveitis (EAU) was induced in B10RIII mice by immunization of interphotoreceptor retinoid binding protein (IRBP; peptide sequence 161-180) or in C57BL/6 (B6) mice by transfer of activated T cells specific for IRBP1-20. The animals were then treated with and without the BLT1 receptor antagonist, CP105696, at the disease onset after immunization or at day 0 or day 6 after T-cell transfer. EAU was also induced in wild-type B6 (WT) and BLT1-deficient (BLT1-/-) mice by reciprocal transfer of the T cells from B6 to BLT1-deficient mice and vise versa. Clinical signs of inflammation and ocular histology were compared. The chemotactic activity of LTB4 on naïve and IRBP-specific autoreactive T cells as well as effector leukocytes was examined.

Results: The treatment of CP105696, greatly reduced the intensity of ongoing disease. IRBP1-20-specific T cells derived from wild-type B6 mice induced only mild uveitis in syngeneic BLT1-deficient mice and that IRBP1-20-specific T cells derived from BLT1-/- mice induced milder disease in wild-type B6 mice than those derived from wild-type B6 mice, suggesting that expression of the LTB4 receptor on both activated autoreactive T cells and effector leukocytes was necessary for ocular inflammation to occur. Consistent with these data, transfer of autoreactive T cells from B6 mice to 5-lipoxygenase-deficient (5-LO-/-) mice, which have a functional defect in LTB4 expression, also failed to induce uveitis in the recipient mice.

Conclusions: The results demonstrate a critical role for LTB4 in ocular inflammation and in the development and progression of EAU and suggest a new potential target for therapeutic intervention in this disease.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adoptive Transfer
  • Animals
  • Arachidonate 5-Lipoxygenase / deficiency
  • Autoimmune Diseases / immunology
  • Autoimmune Diseases / pathology
  • Autoimmune Diseases / prevention & control*
  • Benzopyrans / pharmacology*
  • Carboxylic Acids / pharmacology*
  • Cells, Cultured
  • Chemotaxis, Leukocyte
  • Disease Models, Animal
  • Eye Proteins / immunology
  • Female
  • Immunization
  • Leukotriene B4 / physiology*
  • Lymphocyte Activation
  • Mice
  • Mice, Inbred BALB C
  • Mice, Knockout
  • Peptide Fragments / immunology
  • Purinergic P2 Receptor Antagonists*
  • Receptors, Leukotriene B4 / antagonists & inhibitors*
  • Receptors, Leukotriene B4 / metabolism
  • Receptors, Purinergic P2 / metabolism
  • Retinol-Binding Proteins / immunology
  • T-Lymphocytes / immunology
  • Uveitis / immunology
  • Uveitis / pathology
  • Uveitis / prevention & control*

Substances

  • Benzopyrans
  • Carboxylic Acids
  • Eye Proteins
  • Ltb4r1 protein, mouse
  • Peptide Fragments
  • Purinergic P2 Receptor Antagonists
  • Receptors, Leukotriene B4
  • Receptors, Purinergic P2
  • Retinol-Binding Proteins
  • interstitial retinol-binding protein
  • Leukotriene B4
  • Arachidonate 5-Lipoxygenase
  • CP 105696