CDC25B phosphorylation by p38 and MK-2

Cell Cycle. 2006 Aug;5(15):1649-53. doi: 10.4161/cc.5.15.3006. Epub 2006 Aug 1.

Abstract

CDC25B is one of the three human phosphatases that are involved in the control of the activation of cyclin-dependent kinases. CDC25B participates in regulating entry into mitosis and appears to play a key role in the checkpoint response to DNA injury. CDC25B has been reported to be regulated by a number of kinases and controversial evidence suggests that it is phosphorylated by p38SAPK and/or MAPKAP kinase-2. In this report, we clarify this issue using an approach combining mass spectrometry and the use of specific antibodies against phosphorylated CDC25B residues. We report that MAPKAP kinase-2 phosphorylates CDC25B on multiple sites including S169, S323, S353 and S375, while p38SAPK phosphorylates CDC25B on S249. We show that the S323-phosphorylated form of CDC25B is detected at the centrosome during a normal cell cycle. Since most of these sites are also phosphorylated by several other kinases, our observations highlight the difficulty in characterizing and understanding in vivo phosphorylation patterns.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Antibodies, Phospho-Specific / immunology
  • Cell Cycle Proteins / chemistry
  • Cell Cycle Proteins / metabolism*
  • Enzyme Activation
  • HeLa Cells
  • Humans
  • Intracellular Signaling Peptides and Proteins
  • Mass Spectrometry
  • Molecular Sequence Data
  • Phosphopeptides / metabolism
  • Phosphorylation
  • Phosphoserine / metabolism
  • Protein Serine-Threonine Kinases / metabolism*
  • cdc25 Phosphatases / chemistry
  • cdc25 Phosphatases / metabolism*
  • p38 Mitogen-Activated Protein Kinases / metabolism*

Substances

  • Antibodies, Phospho-Specific
  • Cell Cycle Proteins
  • Intracellular Signaling Peptides and Proteins
  • Phosphopeptides
  • Phosphoserine
  • MAP-kinase-activated kinase 2
  • Protein Serine-Threonine Kinases
  • p38 Mitogen-Activated Protein Kinases
  • CDC25B protein, human
  • cdc25 Phosphatases