Non-selective cation channel on pancreatic duct cells

Biochim Biophys Acta. 1990 Nov 2;1029(1):33-42. doi: 10.1016/0005-2736(90)90433-o.

Abstract

We have identified a non-selective cation channel on pancreatic duct cells. These epithelial cells secrete the bicarbonate ions found in pancreatic juice; a process controlled by the hormone secretin, which uses cyclic AMP as an intracellular messenger. The non-selective channel is located on both apical and basolateral plasma membranes of the duct cell, is equally permeable to sodium and potassium, and has a linear I/V relationship with a single-channel conductance of about 25 pS. Channel opening requires the presence of 1 microM Ca2+ on the cytoplasmic face of the membrane, and is also increased by depolarization. Intracellular ATP, ADP, magnesium, and a rise in pH all decreased channel activity. The channel was not affected by 10 mM TEA, 1 mM Ba2+ or 0.5 mM decamethonium applied to the cytoplasmic face of the membrane, but 0.5 mM quinine caused a flickering block which was more pronounced at depolarizing potentials. We observed the channel only rarely in cell-attached patches on unstimulated duct cells, and acute exposure to stimulants did not cause channel activation. However, after prolonged stimulation, the proportion of cell-attached patches containing active channels was increased 9-fold. The role of this channel in pancreatic duct cell function remains to be elucidated.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenosine Diphosphate / pharmacology
  • Adenosine Triphosphate / pharmacology
  • Animals
  • Calcium / pharmacology
  • Cell Membrane / chemistry
  • Cell Membrane / drug effects
  • Cell Membrane / metabolism
  • Cyclic AMP / metabolism
  • Epithelium / drug effects
  • Epithelium / metabolism
  • Hydrogen-Ion Concentration
  • Ion Channels / chemistry*
  • Ion Channels / drug effects
  • Ion Channels / metabolism
  • Magnesium / pharmacology
  • Membrane Potentials / drug effects
  • Pancreas / chemistry*
  • Pancreas / cytology
  • Pancreas / drug effects
  • Pancreas / metabolism
  • Quinine / pharmacology
  • Rats
  • Second Messenger Systems
  • Secretin / pharmacology

Substances

  • Ion Channels
  • Secretin
  • Adenosine Diphosphate
  • Adenosine Triphosphate
  • Quinine
  • Cyclic AMP
  • Magnesium
  • Calcium