HER2/Neu (ErbB2) signaling to Rac1-Pak1 is temporally and spatially modulated by transforming growth factor beta

Cancer Res. 2006 Oct 1;66(19):9591-600. doi: 10.1158/0008-5472.CAN-06-2071.

Abstract

In HER2 (ErbB2)-overexpressing cells, transforming growth factor beta (TGF-beta), via activation of phosphoinositide-3 kinase (PI3K), recruits actin and actinin to HER2, which then colocalizes with Vav2, activated Rac1, and Pak1 at cell protrusions. This results in prolonged Rac1 activation, enhanced motility and invasiveness, Bad phosphorylation, uncoupling of Bad/Bcl-2, and enhanced cell survival. The recruitment of the HER2/Vav2/Rac1/Pak1/actin/actinin complex to lamellipodia was abrogated by actinin siRNAs, dominant-negative (dn) p85, gefitinib, and dn-Rac1 or dn-Pak1, suggesting that the reciprocal interplay of PI3K, HER2 kinase, and Rac GTPases with the actin cytoskeleton is necessary for TGF-beta action in oncogene-overexpressing cells. Thus, by recruiting the actin skeleton, TGF-beta "cross-links" this signaling complex at cell lamellipodia; this prolongs Rac1 activation and increases metastatic properties and survival of HER2-overexpressing cells.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Actinin / physiology
  • Actins / physiology
  • Adenocarcinoma / pathology
  • Animals
  • Breast Neoplasms / pathology
  • Cell Line, Tumor / metabolism
  • Cell Line, Tumor / ultrastructure
  • Female
  • Humans
  • Mammary Neoplasms, Experimental / pathology
  • Mice
  • Mice, Transgenic
  • Neoplasm Metastasis / physiopathology*
  • Neuropeptides / genetics
  • Neuropeptides / physiology*
  • Phosphatidylinositol 3-Kinases / physiology
  • Phosphoinositide-3 Kinase Inhibitors
  • Protein Serine-Threonine Kinases / genetics
  • Protein Serine-Threonine Kinases / physiology*
  • Proto-Oncogene Proteins c-vav / physiology
  • Pseudopodia / physiology*
  • Pseudopodia / ultrastructure
  • Receptor, ErbB-2 / antagonists & inhibitors
  • Receptor, ErbB-2 / genetics
  • Receptor, ErbB-2 / physiology*
  • Recombinant Fusion Proteins / physiology
  • Signal Transduction / physiology
  • Transforming Growth Factor beta1 / genetics
  • Transforming Growth Factor beta1 / physiology*
  • p21-Activated Kinases
  • rac GTP-Binding Proteins / genetics
  • rac GTP-Binding Proteins / physiology*
  • rac1 GTP-Binding Protein / genetics
  • rac1 GTP-Binding Protein / physiology*

Substances

  • Actins
  • Neuropeptides
  • Phosphoinositide-3 Kinase Inhibitors
  • Proto-Oncogene Proteins c-vav
  • RAC1 protein, human
  • Rac1 protein, mouse
  • Recombinant Fusion Proteins
  • Tgfb1 protein, mouse
  • Transforming Growth Factor beta1
  • VAV2 protein, human
  • Vav2 protein, mouse
  • Actinin
  • ERBB2 protein, human
  • Erbb2 protein, mouse
  • Receptor, ErbB-2
  • PAK1 protein, human
  • Pak1 protein, mouse
  • Protein Serine-Threonine Kinases
  • p21-Activated Kinases
  • rac GTP-Binding Proteins
  • rac1 GTP-Binding Protein