N-acetyl-cysteine protects liver from apoptotic death in an animal model of fulminant hepatic failure

Apoptosis. 2006 Nov;11(11):1945-57. doi: 10.1007/s10495-006-0090-0.

Abstract

Background: This work was undertaken to investigate whether treatment with N-acetyl-cysteine (NAC) prevents oxidative stress and inhibits the apoptotic pathways in an animal model of fulminant hepatic failure.

Methods: Rabbits were experimentally infected with 2x10(4) hemagglutination units of a rabbit hemorrhagic disease virus isolate.

Results: The spontaneous mortality rate of infected animals was 67% at 36 h post infection (pi) and 90% at 48 h pi. This percentage decreased significantly in animals receiving an i.p. injection of NAC (150 mg/kg body way/daily), for 7 days prior to infection. From 36 h pi marked increases were detected in blood levels of transaminases, lactate dehydrogenase, bilirubin and the oxidised/reduced glutathione ratio. All these effects were significantly prevented by NAC treatment. The Bax to Bcl-2 relative expression, the expression of FasL, cytochrome c and PARP-1, and the activity of caspase 3 were significantly increased at 36 and 48 h pi in infected animals. These changes were markedly reduced in animals treated with NAC, with the exception of FasL.

Conclusion: Our results suggest a potential hepatoprotective role of NAC in fulminant hepatic failure, mediated partially through the modulation of the intrinsic pathway of apoptosis.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylcysteine / metabolism
  • Acetylcysteine / pharmacology*
  • Animals
  • Animals, Inbred Strains
  • Antioxidants / metabolism
  • Antioxidants / pharmacology*
  • Apoptosis*
  • Caliciviridae Infections / metabolism
  • Caliciviridae Infections / pathology
  • Disease Models, Animal
  • Hemorrhagic Disease Virus, Rabbit / physiology
  • Hepatocytes / pathology*
  • Hepatocytes / virology
  • Liver / metabolism
  • Liver / pathology*
  • Liver / virology
  • Liver Failure, Acute / metabolism*
  • Liver Failure, Acute / pathology
  • Oxidative Stress / drug effects*
  • Rabbits

Substances

  • Antioxidants
  • Acetylcysteine