Urotensin-II and its receptor (UT-R) are expressed in rat brain endothelial cells, and urotensin-II via UT-R stimulates angiogenesis in vivo and in vitro

Int J Mol Med. 2006 Dec;18(6):1107-12.

Abstract

Urotensin-II (UII), along its receptor UT-R, is widely expressed in the cardiovascular system, where it exerts regulatory actions under both physiological and pathological conditions. Real-time PCR and immunocytochemistry demonstrated the expression of UII and UT-R as mRNA and protein in rat neuromicrovascular endothelial cells (NECs). UII did not affect the proliferation rate of cultured NECs, but exerted a strong angiogenic action in both an in vitro assay on Matrigel and an in vivo assay on chorioallantoic membrane. The angiogenic effect of UII was similar to that of FGF-2, and was abolished by the UT-R antagonist Palosuran. Collectively, our findings allow us to include UII in the group of cytokines (e.g. endothelin-1 and adrenomedullin), which are expressed in endothelial cells and exert a pro-angiogenic effect acting in an autocrine-paracrine manner.

MeSH terms

  • Animals
  • Brain / cytology*
  • Cell Division
  • Cells, Cultured
  • Chick Embryo
  • Chorioallantoic Membrane / blood supply*
  • Chorioallantoic Membrane / drug effects
  • Endothelial Cells / cytology
  • Endothelial Cells / metabolism*
  • Endothelial Cells / physiology
  • Endothelium, Vascular / cytology
  • Immunohistochemistry
  • Immunomagnetic Separation
  • In Vitro Techniques
  • Male
  • Neovascularization, Physiologic / drug effects*
  • Rats
  • Rats, Sprague-Dawley
  • Receptors, G-Protein-Coupled / metabolism*
  • Reverse Transcriptase Polymerase Chain Reaction
  • Time Factors
  • Urotensins / metabolism*
  • Urotensins / pharmacology*

Substances

  • Receptors, G-Protein-Coupled
  • Urotensins
  • urotensin II