Vibrio extracellular protease with prothrombin activation and fibrinolytic activities

Int J Mol Med. 2007 Jan;19(1):157-63.

Abstract

A 36 kDa extracellular metalloprotease (designated to as vEP-MO6) was purified and characterized from Vibrio vulnificus sp. strain MO6 24/0. vEP-MO6 cleaved azocasein and a few other proteins such as prothrombin, plasminogen, fibrinogen and Factor Xa, which are associated with the blood coagulation pathway. The enzyme activity of vEP-MO6 was inhibited by EDTA, which was reversed by the addition of excess divalent cations. vEP-MO6 showed little or no activity toward various chromogenic substrates that are specific for other proteases. The cleavage of prothrombin by vEP-MO6 produced active thrombin, as revealed by an activity assay with thrombin-specific chromogenic substrate and Western blot analysis with anti-thrombin antibody. The enzyme also actively hydrolyzed fibrin polymer as well as the cross-linked fibrin. These results suggest that vEP-MO6 is a prothrombin-activating and cross-linked fibrin-degrading enzyme belonging to the metalloprotease family.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Chelating Agents / pharmacology
  • Enzyme Activation
  • Fibrin / metabolism
  • Fibrinolysis*
  • Metalloproteases / antagonists & inhibitors
  • Metalloproteases / genetics
  • Metalloproteases / isolation & purification
  • Metalloproteases / physiology*
  • Metals / pharmacology
  • Molecular Sequence Data
  • Protease Inhibitors / pharmacology
  • Prothrombin / metabolism*
  • Sequence Homology, Amino Acid
  • Vibrio vulnificus / enzymology*
  • Vibrio vulnificus / genetics

Substances

  • Chelating Agents
  • Metals
  • Protease Inhibitors
  • Prothrombin
  • Fibrin
  • Metalloproteases