Signal transducer and activator of transcription 5b promotes mucosal tolerance in pediatric Crohn's disease and murine colitis

Am J Pathol. 2006 Dec;169(6):1999-2013. doi: 10.2353/ajpath.2006.060186.

Abstract

Growth hormone (GH) regulates anabolic metabolism via activation of the STAT5b transcription factor and reduces mucosal inflammation in colitis. Peroxisome proliferator-activated receptor (PPAR) gamma suppresses mucosal inflammation and is regulated by GH through STAT5b. We hypothesized that the GH:STAT5b axis influences susceptibility to colitis via regulation of local PPARgamma abundance. Colon biopsies from children with newly diagnosed Crohn's disease (CD) and controls were exposed to GH in short-term organ culture. Trinitrobenzene sulfonic acid (TNBS) administration was used to induce colitis in STAT5b-deficient mice and wild-type controls, with and without rosiglitazone pretreatment. GH receptor, STAT5b, PPARgamma, and nuclear factor kappaB activation and expression were determined. Epithelial cell GH receptor expression and GH-dependent STAT5b activation and PPARgamma expression were reduced in CD colon. STAT5b-deficient mice exhibited reduced basal PPARgamma nuclear abundance and developed more severe proximal colitis after TNBS administration. This was associated with a significant increase in mucosal nuclear factor kappaB activation at baseline and after TNBS administration. Rosiglitazone ameliorated colitis in wild-type mice but not STAT5b-deficient mice. GH-dependent STAT5b activation is impaired in affected CD colon and contributes to chronic mucosal inflammation via down-regulation of local PPARgamma expression. Therapeutic activation of the GH:STAT5b axis therefore represents a novel target for restoring both normal anabolic metabolism and mucosal tolerance in CD.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Carrier Proteins / metabolism
  • Child
  • Colitis / therapy*
  • Colon / metabolism
  • Colon / pathology*
  • Crohn Disease / metabolism*
  • Epithelial Cells / metabolism
  • Female
  • Genetic Predisposition to Disease
  • Humans
  • Hypoglycemic Agents / pharmacology
  • Intestinal Mucosa / physiology*
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mucous Membrane / cytology
  • Mucous Membrane / metabolism
  • NF-kappa B / metabolism
  • PPAR gamma / metabolism*
  • Rosiglitazone
  • STAT5 Transcription Factor / genetics
  • STAT5 Transcription Factor / metabolism*
  • STAT5 Transcription Factor / physiology
  • Signal Transduction
  • Thiazolidinediones / pharmacology
  • Trinitrobenzenesulfonic Acid / administration & dosage

Substances

  • Carrier Proteins
  • Hypoglycemic Agents
  • NF-kappa B
  • PPAR gamma
  • STAT5 Transcription Factor
  • STAT5B protein, human
  • Thiazolidinediones
  • Rosiglitazone
  • Trinitrobenzenesulfonic Acid
  • somatotropin-binding protein