Effect of acetyl 11-keto beta-boswellic acid on metastatic growth factor responsible for angiogenesis

Vascul Pharmacol. 2007 May;46(5):333-7. doi: 10.1016/j.vph.2006.09.008. Epub 2006 Nov 10.

Abstract

Basic fibroblast growth factor (bFGF), a metastatic growth factor is known to be one of the promoting factors in the tumor induced angiogenesis. The antiangiogenic activity of acetyl 11-keto beta-boswellic acid was screened against bFGF-induced angiogenesis using in-vivo Matrigel Plug Assay. Histological & colorimetric examination confirmed that numerous blood vessels were present in Matrigel+bFGF group in comparison to Matrigel alone treated mice. Acetyl 11-keto beta-boswellic acids (10 mg/kg/d) inhibited the Matrigel+bFGF-induced angiogenesis significantly (P<0.01) in contrast to anti-inflammatory agent indomethacin (10 mg/kg/d) and alkylating agent cyclophosphamide (10 mg/kg/d).

MeSH terms

  • Angiogenesis Inhibitors / pharmacology*
  • Angiogenesis Inhibitors / therapeutic use
  • Animals
  • Antineoplastic Agents, Alkylating / pharmacology
  • Collagen
  • Cyclooxygenase Inhibitors / pharmacology
  • Cyclophosphamide / pharmacology
  • Disease Models, Animal
  • Drug Combinations
  • Fibroblast Growth Factor 2
  • Indomethacin / pharmacology
  • Laminin
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Neovascularization, Pathologic / chemically induced
  • Neovascularization, Pathologic / pathology
  • Neovascularization, Pathologic / prevention & control*
  • Proteoglycans
  • Reproducibility of Results
  • Subcutaneous Tissue / blood supply*
  • Triterpenes / pharmacology*
  • Triterpenes / therapeutic use

Substances

  • Angiogenesis Inhibitors
  • Antineoplastic Agents, Alkylating
  • Cyclooxygenase Inhibitors
  • Drug Combinations
  • Laminin
  • Proteoglycans
  • Triterpenes
  • acetyl-11-ketoboswellic acid
  • Fibroblast Growth Factor 2
  • matrigel
  • Cyclophosphamide
  • Collagen
  • Indomethacin