Novel chitosan derivative nanoparticles enhance the immunogenicity of a DNA vaccine encoding hepatitis B virus core antigen in mice

J Gene Med. 2007 Apr;9(4):253-64. doi: 10.1002/jgm.1017.

Abstract

Background: Chitosan has been shown to possess useful properties such as non-toxicity, high biocompatibility and non-antigenicity that offer advantages for vaccine delivery systems. In this study, we prepared novel chitosan derivative nanoparticles as DNA vaccine carriers and the potential and mechanism of the DNA-nanoparticle complexes in inducing augmented immune responses were explored.

Methods: The pVAX(HBc)DNA-nanoparticle complexes as vaccine delivery systems were studied in several aspects: the protection against DNase I degradation was measured by an in vitro inhibition assay; the sustained expression of the plasmid in vivo was determined by RT-PCR; the elevated uptake efficiency by phagocytes was observed with confocal microscopy; the biocompatibility was evaluated by cytotoxicity and histology assay; the complexes were administrated to C57BL/6 mice and the humoral and cellular immune responses were evaluated by ELISA, IFN-gamma production and cytolytic T lymphocyte (CTL)-specific lysis assay.

Results: The remaining relative activity of DNase I after inhibition varied from 32.3% to 77.6%. The complexes were observed with higher uptake efficiency by phagocytes than naked DNA. Three types of nanoparticles did not induce significant cytotoxicity at concentrations<or=400 microg/ml. No specific histological alteration related to the injection of the complexes was observed. The formulations of DNA-nanoparticle complexes significantly enhanced the immunogenicity in several parameters: elevated antibody production, higher level of IFN-gamma secretion, and augmented specific cell lysis.

Conclusions: This study demonstrated the potential of the novel chitosan derivative nanoparticles for safe and effective DNA vaccine delivery.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Line, Tumor
  • Chitosan* / chemistry
  • Chitosan* / immunology
  • Deoxyribonuclease I / metabolism
  • Drug Carriers*
  • Drug Delivery Systems
  • Hepatitis B / immunology
  • Hepatitis B / prevention & control
  • Hepatitis B Core Antigens / genetics
  • Hepatitis B Core Antigens / immunology*
  • Humans
  • Immunity / physiology
  • Mice
  • Mice, Inbred C57BL
  • Muscle, Skeletal / cytology
  • Nanoparticles*
  • Vaccines, DNA / immunology*

Substances

  • Drug Carriers
  • Hepatitis B Core Antigens
  • Vaccines, DNA
  • Chitosan
  • Deoxyribonuclease I